Synthesis of tacrine-lophine hybrids via one-pot four component reaction and biological evaluation as acetyl- and butyrylcholinesterase inhibitors
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چکیده
منابع مشابه
Microwave-assisted Synthesis of Acridine-1,8(2H,5H)-diones via a One-pot, Three Component Reaction
A new and improved protocol for the synthesis, in good to excellent yields, of acridine-1,8(2H,5H)-diones is described, involving a one-pot, three component reaction of dimedone, arylglyoxals, and ammonium acetate in water under microwave irradiation.
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ژورنال
عنوان ژورنال: European Journal of Medicinal Chemistry
سال: 2013
ISSN: 0223-5234
DOI: 10.1016/j.ejmech.2013.01.029